SCHEMBL7993417

SCHEMBL7993417

CSc1cccc(N2CCN(CCCCN3C(=O)CS(=O)(=O)C3(C)C)CC2)c1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTR7 P34969 3/20 0.44
KCNH2 Q12809 3/20 0.44
HTR1A P08908 2/20 0.42
HTR6 P50406 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978917 0.86 KCNH2 (0.62) HTR7KCNH2HTR1AHTR6
SCHEMBL7978922 0.86 KCNH2 (0.62) HTR7KCNH2
SCHEMBL7991560 0.83 HTR7 (0.66) HTR7HTR1AHTR6
SCHEMBL7993273 0.81 MAPT (0.46) MAPTMAPK1HTR7KCNH2
Hydrochloric Acid SCHEMBL7997105 0.80 MAPT (0.45) MAPTMAPK1HTR7KCNH2
SCHEMBL7993118 0.73 HTR1A (0.62) HTR7HTR1AHTR6
SCHEMBL7993425 0.72 HTR1A (0.39) HTR7KCNH2HTR1AHTR6
SCHEMBL11377236 0.71 MAPT (0.54) MAPTMAPK1KCNH2
SCHEMBL10518909 0.69 HTR1A (0.54) HTR1A
SCHEMBL17226456 0.69 CHRNA7 (0.59) MAPTMAPK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed