SCHEMBL7994055

SCHEMBL7994055

N#CC1CCN(CCn2cc(-c3cncc(-c4ccsc4)c3)c3c(Cl)cccc32)CC1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 0.56
FLT1 P17948 4/20 0.55
FLT4 P35916 4/20 0.55
CYP2A6 P11509 4/20 0.35
IL1B P01584 2/20 0.32
P2RX7 Q99572 2/20 0.32
TDP2 O95551 1/20 0.32
HTR7 P34969 1/20 0.32
RPS6KB1 P23443 1/20 0.31
AKT1 P31749 1/20 0.31
CXCR3 P49682 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550735 0.89 KDR (0.42) KDRFLT1FLT4IL1BP2RX7
SCHEMBL7547866 0.88 KDR (0.40) KDRFLT1FLT4IL1BP2RX7
SCHEMBL7552023 0.87 KDR (0.40) KDRFLT1FLT4IL1BP2RX7
SCHEMBL7551698 0.87 KDR (0.73) KDRFLT1FLT4CYP2A6IL1B
SCHEMBL7546102 0.86 KDR (0.75) KDRFLT1FLT4CYP2A6
SCHEMBL7990322 0.86 KDR (0.73) KDRFLT1FLT4CYP2A6
SCHEMBL7553661 0.84 SLC6A4 (0.40) KDRFLT1FLT4HTR7
SCHEMBL7557708 0.84 KDR (0.56) KDRFLT1FLT4CYP2A6HTR7
SCHEMBL7976012 0.84 KDR (0.59) KDRFLT1FLT4CYP2A6TDP2
SCHEMBL7976915 0.84 KDR (0.59) KDRFLT1FLT4CYP2A6TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed