SCHEMBL7994283

SCHEMBL7994283

COC(=O)NS(=O)(=O)c1ccccc1-c1ccc(C(=O)C2=CC=CB2)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
RAD52 P43351 1/20 0.34
AGTR1 P30556 1/20 0.34
AGTR2 P50052 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
OXTR P30559 1/20 0.33
MCL1 Q07820 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995486 0.89 ALOX5AP (0.38) ALOX5APFEN1AGTR1AGTR2
SCHEMBL7995536 0.86 ALOX5AP (0.48) ALOX5APFEN1
SCHEMBL7995595 0.83 F10 (0.40) F2PRSS1ALOX5APFEN1
SCHEMBL7995555 0.80 ALOX5AP (0.44) F2PRSS1ALOX5APFEN1TDP1
SCHEMBL7994282 0.78 F2 (0.41) F2PRSS1ALOX5APFEN1AGTR1
SCHEMBL7994030 0.76 F10 (0.36) TDP1
SCHEMBL7994138 0.75 ALOX5AP (0.51) ALOX5APFEN1
SCHEMBL7994014 0.72 ALOX5AP (0.39) ALOX5APFEN1
SCHEMBL8001455 0.72 ALOX5AP (0.45) ALOX5APFEN1
SCHEMBL7984034 0.71 ALOX5AP (0.47) F2PRSS1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810858-A4 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN DU PONT PHARM CO (US) 2000-11-15 EP disclosed
EP-0810858-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-10 EP disclosed
WO-1996020689-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-11 WO disclosed