SCHEMBL7994282

SCHEMBL7994282

COC(=O)NS(=O)(=O)c1ccccc1-c1ccc(C(=O)B2C=CC=C2)c(C)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.41
PRSS1 P07477 1/20 0.41
MCL1 Q07820 2/20 0.36
AGTR1 P30556 1/20 0.35
AGTR2 P50052 1/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995485 0.88 FEN1 (0.41) ALOX5APFEN1
SCHEMBL7995533 0.85 ALOX5AP (0.49) ALOX5APFEN1
SCHEMBL7995594 0.82 F10 (0.42) F2PRSS1MCL1ALOX5APFEN1
SCHEMBL7994283 0.78 F2 (0.38) F2PRSS1MCL1AGTR1AGTR2
SCHEMBL7995553 0.77 ALOX5AP (0.46) F2PRSS1ALOX5APFEN1KDM4E
SCHEMBL10916572 0.76 CASP1 (0.51) AGTR1AGTR2
SCHEMBL7994136 0.73 ALOX5AP (0.54) ALOX5APFEN1
SCHEMBL7128878 0.71 ALOX5AP (0.53) ALOX5APFEN1
SCHEMBL7994011 0.70 ALOX5AP (0.42) ALOX5APFEN1
SCHEMBL7130070 0.70 ALOX5AP (0.55) ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810858-A4 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN DU PONT PHARM CO (US) 2000-11-15 EP disclosed
EP-0810858-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-10 EP disclosed
WO-1996020689-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-11 WO disclosed