SCHEMBL7995486

SCHEMBL7995486

COC(=O)NS(=O)(=O)c1ccccc1-c1ccc(C(=O)C2=CC=CB2)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 15/20 0.38
FEN1 P39748 15/20 0.38
AGTR1 P30556 1/20 0.36
AGTR2 P50052 1/20 0.36
F10 P00742 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7994283 0.89 F2 (0.38) ALOX5APFEN1AGTR1AGTR2
SCHEMBL7994138 0.86 ALOX5AP (0.51) ALOX5APFEN1
SCHEMBL7984034 0.83 ALOX5AP (0.47) ALOX5APFEN1F10
SCHEMBL7995485 0.78 FEN1 (0.41) ALOX5APFEN1
SCHEMBL7995536 0.75 ALOX5AP (0.48) ALOX5APFEN1
SCHEMBL8001509 0.74 AKR1C2 (0.40)
SCHEMBL7994014 0.72 ALOX5AP (0.39) ALOX5APFEN1F10
SCHEMBL10916572 0.70 CASP1 (0.51) AGTR1AGTR2
SCHEMBL8001455 0.69 ALOX5AP (0.45) ALOX5APFEN1
SCHEMBL7994282 0.69 F2 (0.41) ALOX5APFEN1AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810858-A4 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN DU PONT PHARM CO (US) 2000-11-15 EP disclosed
EP-0810858-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-10 EP disclosed
WO-1996020689-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-11 WO disclosed