SCHEMBL7994784

SCHEMBL7994784

C=CCCCCN(C)C(=O)C1C[C@H](Oc2cc(-c3nc(C(F)(F)F)cs3)nc3c(C)c(OC)ccc23)CN1C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
UCHL1 P09936 1/20 0.36
CTSB P07858 1/20 0.34
PPP3CB P16298 1/20 0.34
CTSS P25774 1/20 0.31
ADRB3 P13945 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312962 1.00 UCHL1 (0.36) UCHL1CTSBPPP3CBCTSSADRB3
SCHEMBL312963 1.00 UCHL1 (0.36) UCHL1CTSBPPP3CBCTSSADRB3
SCHEMBL10247253 0.94 UCHL1 (0.36) UCHL1CTSBPPP3CB
SCHEMBL15216085 0.94 UCHL1 (0.36) UCHL1CTSBPPP3CB
SCHEMBL8002444 0.94 UCHL1 (0.36) UCHL1CTSBPPP3CB
SCHEMBL15216171 0.93 CTSB (0.35) CTSBPPP3CBCTSSADRB3ADRA2B
SCHEMBL15026861 0.92 CTSB (0.34) CTSBPPP3CBCTSSADRB3ADRA2B
SCHEMBL10247227 0.91 UCHL1 (0.36) UCHL1CTSBPPP3CB
SCHEMBL8004477 0.89 CTSB (0.32) CTSBPPP3CBCTSS
SCHEMBL313700 0.89 CTSB (0.32) CTSBPPP3CBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed