SCHEMBL8004477

SCHEMBL8004477

C=CCCCCN(C)C(=O)C1C[C@H](Oc2cc(-c3nc(C(F)(F)F)cs3)nc3c(C)c(OC)ccc23)CN1C(=O)n1ccnc1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.32
PPP3CB P16298 1/20 0.32
CTSS P25774 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL313700 1.00 CTSB (0.32) CTSBPPP3CBCTSS
SCHEMBL8005334 0.94 CTSB (0.32) CTSBPPP3CB
SCHEMBL12356928 0.94 CTSB (0.32) CTSBPPP3CB
SCHEMBL12369706 0.92 CTSS (0.32) CTSBPPP3CBCTSS
SCHEMBL10247430 0.92
SCHEMBL15216171 0.90 CTSB (0.35) CTSBPPP3CBCTSS
SCHEMBL15026861 0.90 CTSB (0.34) CTSBPPP3CBCTSS
SCHEMBL7994784 0.89 UCHL1 (0.36) CTSBPPP3CBCTSS
SCHEMBL312962 0.89 UCHL1 (0.36) CTSBPPP3CBCTSS
SCHEMBL312963 0.89 UCHL1 (0.36) CTSBPPP3CBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed