SCHEMBL7994824

SCHEMBL7994824

[CH2]CCN1CCC(C#N)(c2ccccc2C#N)CC1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.44
OPRD1 P41143 1/20 0.42
ADRA1A P35348 8/20 0.41
OPRL1 P41146 1/20 0.40
ADRA1D P25100 5/20 0.39
ADRA1B P35368 5/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7668749 0.84 OPRM1 (0.48) OPRM1ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL7702085 0.83 OPRM1 (0.47) OPRM1ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL7664127 0.83 OPRM1 (0.47) OPRM1ADRA1AADRA1DADRA1B
SCHEMBL8010117 0.82 ADRA1A (0.47) OPRM1ADRA1AADRA1DADRA1B
SCHEMBL7668741 0.81 ADRA1A (0.44) OPRM1ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL7664114 0.80 ADRA1A (0.44) OPRM1ADRA1AADRA1DADRA1B
SCHEMBL7840973 0.80 OPRM1 (0.66) OPRM1OPRD1ADRA1AOPRL1ADRA1D
SCHEMBL10526389 0.78 TSHR (0.40) OPRM1ADRA1A
SCHEMBL30410927 0.78 TSHR (0.40) OPRM1ADRA1A
SCHEMBL17434404 0.75 NPC1 (0.38) OPRM1ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000025782-A1 DIHYDROPYRIDINONES AND PYRROLINONES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-11 WO claimed
WO-2000025782-A1 DIHYDROPYRIDINONES AND PYRROLINONES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-11 WO disclosed