SCHEMBL7995257

SCHEMBL7995257

COc1cccc(Oc2ccc3c(c2)COB3)c1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
PGR P06401 4/20 0.44
MTNR1B P49286 8/20 0.43
MTNR1A P48039 6/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
AADAT Q8N5Z0 2/20 0.41
LTA4H P09960 1/20 0.41
ACACB O00763 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801556 0.86 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DAADAT
SCHEMBL28176199 0.82 TMEM97 (0.47)
SCHEMBL14748454 0.82 MAOB (0.53) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL14748434 0.81 PDE4A (0.50) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL14748410 0.81 ALDH1A1 (0.54) MTNR1B
SCHEMBL8012418 0.79 MAOA (0.40) PDE4APDE4BPDE4CPDE4D
SCHEMBL8007552 0.78 PDE4A (0.50) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL19622266 0.78 ALDH1A1 (0.47) SMN1; SMN2PDE4APDE4BPDE4CPDE4D
SCHEMBL8007094 0.78 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DLTA4H
SCHEMBL8010793 0.78 ST14 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed