SCHEMBL7995263

SCHEMBL7995263

CNCc1ccc(Oc2ccccc2)c(S(C)(=O)=O)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.48
HTR2A P28223 2/20 0.48
HTR7 P34969 1/20 0.43
KCNQ3 O43525 2/20 0.42
KCNQ2 O43526 2/20 0.42
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TTR P02766 2/20 0.40
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNH2 Q12809 1/20 0.40
PTGS2 P35354 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8004812 0.76 KCNQ3 (0.42) KCNQ3KCNQ2SMN1; SMN2CYP2D6SLC6A3
SCHEMBL9018653 0.76 KCNQ3 (0.40) KCNQ3KCNQ2MAPTLMNACA2
SCHEMBL29625906 0.75 BRD4 (0.46) SMN1; SMN2PTGS2CYP3A4
SCHEMBL28738313 0.75 BRD4 (0.46) SMN1; SMN2PTGS2CYP3A4
SCHEMBL29181894 0.75 MEN1 (0.58) MAPTLMNASMN1; SMN2TTRKDM4E
SCHEMBL8005449 0.72 TTR (0.61) MAPTLMNASMN1; SMN2TTRPTGS2
SCHEMBL7995261 0.72 TTR (0.61) TTRCA2CA4
SCHEMBL8004004 0.72 KCNQ3 (0.39) KCNQ3KCNQ2CYP2D6SLC6A3CA2
SCHEMBL1108585 0.71 KDM4E (0.61) SLC6A4HTR2AMAPTSMN1; SMN2KDM4E
SCHEMBL1351804 0.71 KDM4E (0.62) MAPTSMN1; SMN2KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed