SCHEMBL9018653

SCHEMBL9018653

CNC(=N)N(CS(=O)(=O)O)C(=O)NCc1ccc(Oc2ccccc2)c(S(C)(=O)=O)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 2/20 0.40
KCNQ2 O43526 2/20 0.40
MAPK14 Q16539 2/20 0.38
CA2 P00918 1/20 0.38
CA4 P22748 1/20 0.38
ALDH1A1 P00352 3/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PPARG P37231 3/20 0.33
PPARA Q07869 3/20 0.33
PPARD Q03181 2/20 0.33
ERCC1 P07992 1/20 0.33
ERCC4 Q92889 1/20 0.33
P2RX4 Q99571 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089145 0.81 SLC9A1 (0.39) ERCC1ERCC4
SCHEMBL8004812 0.81 KCNQ3 (0.42) KCNQ3KCNQ2MAPK14CA2CA4
SCHEMBL9018660 0.76 POLB (0.33) KCNQ3KCNQ2CA2CA4ALDH1A1
SCHEMBL7995263 0.76 SLC6A4 (0.48) KCNQ3KCNQ2CA2CA4LMNA
SCHEMBL8004004 0.69 KCNQ3 (0.39) KCNQ3KCNQ2CA2CA4L3MBTL1
SCHEMBL9018656 0.67 POLB (0.37) CA2CA4L3MBTL1P2RX4
SCHEMBL29625910 0.65 IDH1 (0.56) MAPK14CA2P2RX4MAPT
SCHEMBL28738385 0.65 IDH1 (0.56) MAPK14CA2P2RX4MAPT
SCHEMBL7995261 0.65 TTR (0.61) CA2CA4ALDH1A1NPSR1
SCHEMBL9018671 0.64 TTR (0.38) KCNQ3KCNQ2CA2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP claimed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed