SCHEMBL7995476

SCHEMBL7995476

NS(=O)(=O)c1ccccc1-c1ccc(C(=O)B2C=CC=C2)c([N+](=O)[O-])c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F10 P00742 6/20 0.44
CA9 Q16790 3/20 0.39
CA2 P00918 2/20 0.39
SCN9A Q15858 1/20 0.39
ALOX5AP P20292 2/20 0.38
FEN1 P39748 2/20 0.38
ALDH1A1 P00352 3/20 0.37
TRPV1 Q8NER1 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
POLB P06746 1/20 0.37
KCNMA1 Q12791 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7994011 0.84 ALOX5AP (0.42) ALOX5APFEN1
SCHEMBL7995594 0.81 F10 (0.42) F10SCN9AALOX5APFEN1TRPV1
SCHEMBL7995479 0.77 F10 (0.44) F10CA9CA2SCN9AALOX5AP
SCHEMBL5968143 0.74 ALOX5AP (0.51) F10CA9CA2SCN9AALOX5AP
SCHEMBL10864758 0.68 CA1 (0.59) F10CA9CA2SCN9ACA12
SCHEMBL29481486 0.68 CA1 (0.59) F10CA9CA2SCN9ACA12
SCHEMBL4664143 0.68 CA2 (0.55) CA9CA2SCN9AALDH1A1CA12
SCHEMBL28163944 0.67 ALDH1A1 (0.47) CA9CA2SCN9AALDH1A1CYP1A2
SCHEMBL7995533 0.67 ALOX5AP (0.49) ALOX5APFEN1
SCHEMBL7994136 0.66 ALOX5AP (0.54) ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810858-A4 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN DU PONT PHARM CO (US) 2000-11-15 EP disclosed
EP-0810858-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-10 EP disclosed
WO-1996020689-A2 BORONIC ACID AND ESTER INHIBITORS OF THROMBIN THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-11 WO disclosed