SCHEMBL7995531

SCHEMBL7995531

COC(=O)c1cc(C(=O)OC)cc(-c2cc(OC)ccc2Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
KDM4E B2RXH2 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 2/20 0.46
ALDH1A1 P00352 3/20 0.45
SCN10A Q9Y5Y9 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42
EIF4E P06730 1/20 0.41
NR4A2 P43354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995380 0.94 CA1 (0.45) CA1CA2KDM4ECYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8663603 0.83 CYP2D6 (0.47) CYP1A2CYP2D6KMT2AMAPTALDH1A1
SCHEMBL3874099 0.80 CA1 (0.45) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL2409870 0.80 TSHR (0.49) CA1CA2KDM4EMAPTPOLB
SCHEMBL8005356 0.79 MAPT (0.44) KDM4EKMT2AMEN1MAPTALDH1A1
SCHEMBL8005976 0.78 MAPT (0.52) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL13715371 0.77 CA1 (0.49) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL12774551 0.77 CA1 (0.66) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL8818855 0.77 CA12 (0.53) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL2437425 0.76 TSHR (0.49) CA1CA2KDM4EMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017917-A Guanidine derivatives FUJISAWA PHARAMCEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0876338-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-11-11 EP disclosed
WO-1997025310-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-17 WO disclosed