SCHEMBL7995380

SCHEMBL7995380

COC(=O)c1cc(C(=O)O)cc(-c2cc(OC)ccc2Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
KDM4E B2RXH2 2/20 0.44
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PRKAB2 O43741 2/20 0.43
PRKAG1 P54619 2/20 0.43
PRKAA2 P54646 2/20 0.43
PRKAA1 Q13131 2/20 0.43
PRKAG3 Q9UGI9 2/20 0.43
PRKAG2 Q9UGJ0 2/20 0.43
PRKAB1 Q9Y478 2/20 0.43
EIF4E P06730 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7995531 0.94 CA1 (0.50) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL8005356 0.86 MAPT (0.44) KDM4EMEN1KMT2AMAPTTPMT
SCHEMBL8005976 0.85 MAPT (0.52) CA1CA2KDM4ECYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8663603 0.78 CYP2D6 (0.47) CYP1A2CYP2D6KMT2AMAPTSMN1; SMN2
SCHEMBL3874099 0.76 CA1 (0.45) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL56890 0.76 KDM4E (0.55) CA1CA2KDM4EGAAPOLB
SCHEMBL2427192 0.76 CA1 (0.58) CA1CA2KDM4EPRKAB2PRKAG1
SCHEMBL6252554 0.76 ALDH1A1 (0.51) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL2409870 0.75 TSHR (0.49) CA1CA2KDM4EGAAPOLB
SCHEMBL28904089 0.74 KDM4E (0.53) CA1CA2KDM4EGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017917-A Guanidine derivatives FUJISAWA PHARAMCEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0876338-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-11-11 EP disclosed
WO-1997025310-A1 GUANIDINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-07-17 WO disclosed