SCHEMBL7995693

SCHEMBL7995693

Cc1c(Cn2ccnc2[N+](=O)[O-])cccc1OCCCSc1ncccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
CYP2D6 P10635 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
NPC1 O15118 5/20 0.38
RAB9A P51151 5/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
MAPT P10636 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HSD17B10 Q99714 2/20 0.37
POLB P06746 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001628 0.90 GRM2 (0.41) KMT2AMEN1CYP2D6NPC1RAB9A
SCHEMBL7994851 0.86 EGFR (0.33) CYP2D6MAPTHTTLMNATYMP
SCHEMBL7995736 0.85 CYP1A2 (0.43) KMT2AMEN1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL7984644 0.84 TYMP (0.38) KMT2AMEN1CYP2D6CYP2C19NPC1
SCHEMBL8001605 0.83 LMNA (0.42) KMT2ACYP2D6CYP2C19ALDH1A1POLB
SCHEMBL7996140 0.81 KMT2A (0.39) KMT2AMEN1CYP2D6CYP1A2CYP2C9
SCHEMBL7984159 0.81 EGFR (0.31) EGFR
SCHEMBL7994182 0.81 KMT2A (0.40) KMT2AMEN1CYP2D6CYP1A2CYP2C9
SCHEMBL7994293 0.81 NPC1 (0.42) KMT2AMEN1CYP2D6CYP1A2CYP2C9
SCHEMBL7984571 0.79 CYP3A4 (0.43) KMT2ACYP2D6CYP2C19SMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO claimed
WO-2001034578-A1 COMPOUNDS WITH ANTI-HELICOBACTER PYLORI ACTIVITY ASTRAZENECA AB (SE) 2001-05-17 WO disclosed