SCHEMBL7995720

SCHEMBL7995720

CNc1cccc(C(C)=CCCN)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
PARP1 P09874 5/20 0.35
PARP10 Q53GL7 4/20 0.35
PARP14 Q460N5 1/20 0.35
CREBBP Q92793 1/20 0.34
PARP15 Q460N3 1/20 0.34
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
RAB9A P51151 1/20 0.33
NTSR1 P30989 1/20 0.32
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7546895 0.82 MEN1 (0.40) MEN1KMT2AALDH1A1CREBBPMAPT
SCHEMBL27955929 0.78 PTGS1 (0.50) PARP1MAPTRAB9A
SCHEMBL20998077 0.71 MAOA (0.41) MEN1KMT2AALDH1A1PARP1PARP10
SCHEMBL6251424 0.69 MEN1 (0.40) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL6251422 0.69 MEN1 (0.40) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL7768635 0.69 ALDH1A1 (0.66) MEN1KMT2AALDH1A1CREBBPSMN1; SMN2
SCHEMBL8577301 0.69 TDP1 (0.49) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL30478066 0.69 ALDH1A1 (0.66) MEN1KMT2AALDH1A1CREBBPSMN1; SMN2
SCHEMBL14253754 0.68 MEN1 (0.45) MEN1KMT2AALDH1A1MAPTSMN1; SMN2
SCHEMBL21792030 0.68 ALDH1A1 (0.59) MEN1KMT2AALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042274-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-10-11 EP disclosed
WO-2000023418-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-27 WO disclosed