SCHEMBL8005665

SCHEMBL8005665

COc1ccc2c(C)cc(-c3csc(C(F)(F)F)n3)nc2c1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.37
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
RAB9A P51151 5/20 0.35
NPC1 O15118 4/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
ENPP3 O14638 1/20 0.33
ENPP1 P22413 1/20 0.33
PDE4B Q07343 4/20 0.32
PDE4A P27815 2/20 0.32
PDE4C Q08493 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3797063 0.89 GAA (0.37) RORCKDM4EALDH1A1RAB9ANPC1
SCHEMBL8005821 0.89 ALDH1A1 (0.39) RORCKDM4EALDH1A1RAB9ANPC1
SCHEMBL7996164 0.88 RAB9A (0.37) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL7996053 0.82 KDM4E (0.36) RORCKDM4EALDH1A1RAB9ANPC1
SCHEMBL577373 0.78 ALDH1A1 (0.35) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL13090548 0.77 MAPT (0.40) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL15216114 0.77 GAA (0.38) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL15216089 0.77 ALDH1A1 (0.38) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL8135741 0.74 ALDH1A1 (0.39) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL15692157 0.73 RXFP1 (0.45) KDM4EALDH1A1NPC1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed