SCHEMBL8003756

SCHEMBL8003756

COc1ccc2c(N)cc(-c3nc(C(F)(F)F)cs3)nc2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
G6PD P11413 1/20 0.34
PDE4B Q07343 8/20 0.34
PDE4A P27815 3/20 0.34
PDE4C Q08493 3/20 0.34
PDE4D Q08499 3/20 0.34
PDE11A Q9HCR9 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
PTGES O14684 1/20 0.34
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3674311 0.89 PDE4B (0.37) KDM4EALDH1A1PDE4BPDE4APDE4C
SCHEMBL15216086 0.88 PDE4B (0.35) KDM4EALDH1A1PDE4BNPC1RAB9A
SCHEMBL7996051 0.88 KMT2A (0.37) KDM4EALDH1A1PDE4BPDE4APDE4C
SCHEMBL7996053 0.88 KDM4E (0.36) KDM4EALDH1A1PDE4BPDE4APDE4C
SCHEMBL7996056 0.87 SLC2A1 (0.35) KDM4EALDH1A1PDE4BPDE11ANPC1
SCHEMBL313131 0.87 PDE4B (0.36) ALDH1A1PDE4BPDE4APDE4CPDE4D
SCHEMBL8005137 0.84 KDM4E (0.39) KDM4EALDH1A1G6PDNPC1RAB9A
SCHEMBL8005821 0.81 ALDH1A1 (0.39) KDM4EALDH1A1G6PDPDE4BPDE4A
SCHEMBL8006162 0.81 ALDH1A1 (0.37) KDM4EALDH1A1G6PDNPC1RAB9A
SCHEMBL8008384 0.80 ALDH1A1 (0.36) KDM4EALDH1A1G6PDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed