SCHEMBL7997129

SCHEMBL7997129

Clc1ccc2c(C3CNCCN3)csc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.36
HTR2C P28335 6/20 0.36
HTR2B P41595 6/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CNR1 P21554 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
HRH1 P35367 1/20 0.36
KCNH2 Q12809 1/20 0.36
CYP2A6 P11509 4/20 0.35
CHRNB2 P17787 1/20 0.33
CHRNA4 P43681 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993389 0.83 MAPT (0.36) HTR2AHTR2CKCNH2CHRNB2CHRNA4
SCHEMBL7993430 0.81 SLC6A4 (0.40) SLC6A4CYP2A6SMN1; SMN2CA1CA2
Hydrochloric Acid SCHEMBL2957745 0.79 HTR2C (0.39) HTR2AHTR2CHTR2BHTR1AKCNH2
SCHEMBL16165 0.75 HTR2C (0.45) HTR2AHTR2CHTR2BADRB1HTR1A
SCHEMBL1638955 0.75 HTR2C (0.44) HTR2AHTR2CHTR2BADRB1HTR1A
SCHEMBL7997135 0.71 HTR2C (0.37) HTR2AHTR2CHTR2BADRB1HTR1A
SCHEMBL9590723 0.69 ROCK1 (0.40) HTR2AHTR2CHTR2BADRB1HTR1A
SCHEMBL1673686 0.68 HTR3A (0.53) SLC6A2SLC6A4HTR3A
SCHEMBL263978 0.68 HTR3A (0.53) SLC6A2SLC6A4HTR3A
SCHEMBL9591713 0.68 HTR2C (0.33) HTR2AHTR2CHTR2BADRB1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed
US-5136037-A 3-(4-substituted-4-piperazinyl)butyl-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-04 US disclosed
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4933453-A ANTIPSYCHOTIC, ANALGESIC, ANTICONVULSANT, AND ANXIOLYTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-12 US disclosed