SCHEMBL7999300

SCHEMBL7999300

CC(C)C(=O)CCc1ccc(NC(=O)OCc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
TP53 P04637 2/20 0.52
MAPT P10636 2/20 0.52
RAB9A P51151 5/20 0.51
NPC1 O15118 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
KDM1A O60341 2/20 0.51
MAOA P21397 2/20 0.51
MAOB P27338 2/20 0.51
ALDH1A1 P00352 1/20 0.51
TSHR P16473 1/20 0.51
ATM Q13315 1/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.51
MGLL Q99685 1/20 0.50
ROCK2 O75116 1/20 0.50
RCOR1 Q9UKL0 1/20 0.50
RECQL P46063 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21054940 0.85 POLB (0.62) POLBTP53MAPTRAB9ANPC1
SCHEMBL590420 0.82 POLB (0.62) POLBTP53MAPTRAB9ANPC1
SCHEMBL3070644 0.82 POLB (0.56) POLBTP53MAPTRAB9ANPC1
SCHEMBL8867533 0.81 POLB (0.64) POLBTP53MAPTRAB9ANPC1
SCHEMBL3968088 0.81 POLB (0.64) POLBTP53MAPTRAB9ANPC1
SCHEMBL8579394 0.80 SMN1; SMN2 (0.61) POLBTP53MAPTRAB9ANPC1
SCHEMBL13666356 0.80 POLB (0.59) POLBTP53MAPTRAB9ANPC1
SCHEMBL16942604 0.80 POLB (0.62) POLBTP53MAPTRAB9ANPC1
SCHEMBL19682897 0.80 POLB (0.62) POLBTP53MAPTRAB9ANPC1
SCHEMBL23917849 0.79 ALDH1A1 (0.69) POLBTP53MAPTRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
US-5834506-A TREATMENT OF HIV, AIDS; ANTIVIRAL ACTIVITY IMPROVED BY JUDICIOUS PLACEMENT OF POLAR SUBSTITUENTS WARNER-LAMBERT COMPANY (US) 1998-11-10 US disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed