SCHEMBL7999742

SCHEMBL7999742

NS(=O)(=O)c1ccccc1CO[PH](=O)OCc1ccccc1S(N)(=O)=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.42
CA1 P00915 12/20 0.42
CA9 Q16790 10/20 0.42
CA12 O43570 4/20 0.42
CA6 P23280 3/20 0.42
CA5A P35218 3/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
CA5B Q9Y2D0 2/20 0.42
CA14 Q9ULX7 2/20 0.42
CYP2C9 P11712 1/20 0.42
PTGES2 Q9H7Z7 3/20 0.37
LDHA P00338 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19280573 0.79 IDO1 (0.53) CA2CA1CA9CA12CA6
SCHEMBL31726638 0.78 CA2 (0.47) CA2CA1CA9CA12CA6
SCHEMBL574790 0.78 CA2 (0.47) CA2CA1CA9CA12CA6
SCHEMBL1128972 0.75 CA2 (0.51) CA2CA1CA9CA12CA6
SCHEMBL8349565 0.74 CA2 (0.54) CA2CA1CA9CA12CA6
SCHEMBL11046847 0.74 CA2 (0.41) CA2CA1CA9CA12CA6
SCHEMBL27351284 0.73 P2RX4 (0.42) CA2CA1CA9CA12CA6
SCHEMBL6939683 0.73 FDPS (0.38)
SCHEMBL1517165 0.73 IDO1 (0.55) CA2CA9CA12
SCHEMBL731097 0.73 TAAR1 (0.52) CA2CA1CA9CA12CA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288100-B1 SUCH AS PHENYL-(2-PROPYL-1H-BENZIMIDAZOL-5-YL)-METHANONE USEFUL AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION 2001-09-11 US disclosed
EP-0830343-A1 BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-25 EP disclosed
WO-1996039390-A1 BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1996-12-12 WO disclosed