SCHEMBL7999769

SCHEMBL7999769

COc1cc(CN2CCNCC2=O)cc(OC)c1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
HTR6 P50406 1/20 0.41
GAA P10253 2/20 0.40
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
KMT2A Q03164 4/20 0.38
MEN1 O00255 3/20 0.38
PKM P14618 1/20 0.38
GPR183 P32249 1/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
CASP1 P29466 1/20 0.36
CASP4 P49662 1/20 0.36
CASP5 P51878 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20133743 0.85 GAA (0.57) ADRB1GAAKMT2AMEN1ALDH1A1
Hydrochloric Acid SCHEMBL6410332 0.82 FAAH (0.33) TDP1KMT2AMEN1
SCHEMBL18076484 0.78 GAA (0.53) GAAKMT2AMEN1ALDH1A1
SCHEMBL25425946 0.76 QPCT (0.44) ADRB1KMT2AMEN1PKMALDH1A1
SCHEMBL29194592 0.76 PKM (0.46) KMT2AMEN1PKMALDH1A1
SCHEMBL30854970 0.76 QPCT (0.44) ADRB1KMT2AMEN1PKMALDH1A1
SCHEMBL30245048 0.76 PKM (0.46) KMT2AMEN1PKMALDH1A1
SCHEMBL11628726 0.76 ADRB1 (0.56) ADRB1TDP1KMT2AMEN1GPR183
SCHEMBL28830636 0.75 HRH2 (0.38) ADRB1KMT2AMEN1HTR2C
SCHEMBL25426716 0.73 PKM (0.43) KMT2AMEN1PKMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000008005-A2 PIPERAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2000-02-17 WO disclosed