SCHEMBL7999871

SCHEMBL7999871

Cc1nc(-c2cccc(CN3CCN(C(=O)c4ccc(-c5ccccc5)cc4)CC3=O)c2)no1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 3/20 0.48
CYP46A1 Q9Y6A2 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HCRTR1 O43613 4/20 0.46
HCRTR2 O43614 4/20 0.46
LMNA P02545 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
RECQL P46063 1/20 0.46
KMT2A Q03164 1/20 0.46
MET P08581 1/20 0.44
PLA2G2A P14555 2/20 0.42
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
DAO P14920 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003104 0.92 MGLL (0.46) MGLLCYP46A1HRH3HCRTR1HCRTR2
SCHEMBL7999939 0.92 MGLL (0.52) MGLLCYP46A1HRH3KMT2APLA2G2A
SCHEMBL7997634 0.91 NPC1 (0.45) MGLLCYP46A1HRH3HCRTR1HCRTR2
SCHEMBL7996195 0.85 NPC1 (0.42) MGLLCYP46A1HRH3LMNAMAPT
SCHEMBL7996342 0.84 HCRTR1 (0.47) HRH3HCRTR1HCRTR2LMNAALDH1A1
SCHEMBL7999739 0.84 NPC1 (0.47) MGLLCYP46A1HRH3LMNAPLA2G2A
SCHEMBL7996149 0.82 HCRTR1 (0.46) HCRTR1HCRTR2LMNAALDH1A1MAPT
SCHEMBL7999727 0.79 HCRTR1 (0.46) HRH3HCRTR1HCRTR2LMNAALDH1A1
SCHEMBL7074772 0.79 MGLL (0.66) MGLLLMNAALDH1A1MAPTMEN1
SCHEMBL7999778 0.77 SLC2A1 (0.43) HRH3HCRTR1HCRTR2LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000008005-A2 PIPERAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2000-02-17 WO disclosed