SCHEMBL7997634

SCHEMBL7997634

Cc1nc(-c2cccc(CN3CCN(C(=O)c4ccc5ccccc5c4)CC3=O)c2)no1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.45
HCRTR1 O43613 4/20 0.45
HCRTR2 O43614 4/20 0.45
CYP46A1 Q9Y6A2 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
MET P08581 1/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MGLL Q99685 1/20 0.41
GRM5 P41594 1/20 0.40
RHOA P61586 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SPHK2 Q9NRA0 1/20 0.40
SPHK1 Q9NYA1 1/20 0.40
LMNA P02545 1/20 0.40
AKR1C1 Q04828 1/20 0.39
DAO P14920 1/20 0.39
PLA2G2A P14555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7996195 0.92 NPC1 (0.42) NPC1CYP46A1HRH3HPGDTSHR
SCHEMBL7999871 0.91 MGLL (0.48) HCRTR1HCRTR2CYP46A1HRH3MET
SCHEMBL7999739 0.91 NPC1 (0.47) NPC1CYP46A1HRH3HPGDTSHR
SCHEMBL8003104 0.87 MGLL (0.46) HCRTR1HCRTR2CYP46A1HRH3MGLL
SCHEMBL7999939 0.83 MGLL (0.52) CYP46A1HRH3MGLLPLA2G2A
SCHEMBL7076687 0.78 TSHR (0.59) NPC1HPGDTSHRMGLLLMNA
SCHEMBL7996342 0.77 HCRTR1 (0.47) HCRTR1HCRTR2HRH3METTSHR
SCHEMBL7996221 0.77 PLA2G2A (0.42) HCRTR1HCRTR2HRH3TSHRSPHK2
SCHEMBL7071609 0.77 NPC1 (0.65) NPC1HPGDTSHRMGLLL3MBTL1
SCHEMBL7999722 0.76 ALDH1A1 (0.45) HCRTR1HCRTR2HRH3TSHRSPHK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000008005-A2 PIPERAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2000-02-17 WO disclosed