SCHEMBL7999874

SCHEMBL7999874

COC(=O)CC(=O)CC(O)(CCc1ccc(O)cc1)C1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MIF P14174 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM4E B2RXH2 2/20 0.35
F13A1 P00488 1/20 0.35
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
EPHX2 P34913 1/20 0.34
MEN1 O00255 1/20 0.34
EPHX1 P07099 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13964139 0.90 RAB9A (0.40) NPC1RAB9ACYP1A2CYP3A4CYP2D6
SCHEMBL13964064 0.89 SSTR3 (0.41) RAB9A
SCHEMBL3437561 0.79 PTGDR (0.33) RAB9AHPGDEPHX2MEN1EPHX1
SCHEMBL13963700 0.77 CA1 (0.42) MEN1KMT2A
SCHEMBL13964128 0.77 ALDH1A1 (0.32) HPGDALDH1A1
SCHEMBL13964137 0.76 MAPT (0.37) HPGDALDH1A1MAPT
SCHEMBL13964266 0.74 SCN9A (0.40) CYP3A4CYP2C9CYP2C19EPHX2
SCHEMBL3988297 0.73 GABRP (0.40) NPC1MEN1KMT2A
SCHEMBL5880783 0.72 NPC1 (0.43) NPC1RAB9AHPGDKDM4EEPHX2
SCHEMBL3988475 0.72 GABRP (0.39) MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046355-A TOLUENE-4-THIOSULFONIC ACID S-ESTERS AS CHEMICAL INTERMEDIATES FOR VIRICIDES AND ASPARTYL PROTEASE INHIBITORS; AIDS WARNER-LAMBERT COMPANY (US) 2000-04-04 US disclosed
EP-0935597-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1999-08-18 EP disclosed
US-5834506-A TREATMENT OF HIV, AIDS; ANTIVIRAL ACTIVITY IMPROVED BY JUDICIOUS PLACEMENT OF POLAR SUBSTITUENTS WARNER-LAMBERT COMPANY (US) 1998-11-10 US disclosed
WO-1998019997-A2 DIHYDROPYRONES WITH IMPROVED ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed