SCHEMBL8000685

SCHEMBL8000685

COc1ccc(-n2nnc(C)n2)cc1/C=C/CC(C)(C)Cc1csc(C)n1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
RAB9A P51151 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
HCRTR2 O43614 1/20 0.32
CYP1A2 P05177 1/20 0.30
SLC5A7 Q9GZV3 1/20 0.30
METAP2 P50579 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009912 0.88 ALDH1A1 (0.38) ALDH1A1RAB9AL3MBTL1HCRTR2CYP1A2
SCHEMBL8008288 0.86 ALDH1A1 (0.31) ALDH1A1RAB9A
SCHEMBL8005747 0.86 ALDH1A1 (0.37) ALDH1A1RAB9AL3MBTL1CYP1A2SLC5A7
SCHEMBL7999092 0.84 ALDH1A1 (0.36) ALDH1A1RAB9AL3MBTL1CYP1A2SLC5A7
SCHEMBL7998586 0.84 ALDH1A1 (0.35) ALDH1A1RAB9AL3MBTL1CYP1A2SLC5A7
SCHEMBL10260150 0.81 CSF1R (0.30)
SCHEMBL8008671 0.81 ALDH1A1 (0.36) ALDH1A1RAB9AL3MBTL1HCRTR2CYP1A2
SCHEMBL8000689 0.81 ENPP2 (0.32)
SCHEMBL10292899 0.79
SCHEMBL8009669 0.79 ALDH1A1 (0.35) ALDH1A1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed