SCHEMBL8008671

SCHEMBL8008671

COc1ccc(-n2nnc(C)n2)cc1CCCC(C)(C)Cc1csc(C)n1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
HCRTR2 O43614 1/20 0.33
USP2 O75604 1/20 0.32
PKM P14618 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP1A2 P05177 1/20 0.31
SLC5A7 Q9GZV3 1/20 0.31
METAP2 P50579 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
SLC6A4 P31645 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7999097 0.88 ALDH1A1 (0.39) ALDH1A1RAB9AL3MBTL1HCRTR2USP2
SCHEMBL8016004 0.88 ALDH1A1 (0.39) ALDH1A1RAB9AL3MBTL1HCRTR2USP2
SCHEMBL7999100 0.88 ALDH1A1 (0.39) ALDH1A1RAB9AL3MBTL1HCRTR2USP2
SCHEMBL7999173 0.88 ALDH1A1 (0.39) ALDH1A1RAB9AL3MBTL1HCRTR2USP2
SCHEMBL8008285 0.86 ALDH1A1 (0.33) ALDH1A1RAB9A
SCHEMBL8000685 0.81 ALDH1A1 (0.35) ALDH1A1RAB9AL3MBTL1HCRTR2CYP1A2
SCHEMBL10260245 0.80 CSF1R (0.31)
SCHEMBL8014614 0.79 ENPP2 (0.32)
SCHEMBL10292822 0.79 CSF1R (0.30)
SCHEMBL8008299 0.79 TACR1 (0.38) ALDH1A1RAB9AL3MBTL1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed