SCHEMBL8002147

SCHEMBL8002147

COc1cc2c(c(C)c1C)C(=O)C(O)(O)C2=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 16/20 0.65
CA2 P00918 16/20 0.65
CA7 P43166 16/20 0.65
CA9 Q16790 16/20 0.65
CA4 P22748 2/20 0.45
EPHX2 P34913 2/20 0.38
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
RECQL P46063 1/20 0.35
BACE1 P56817 1/20 0.35
EHMT2 Q96KQ7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP3A4 P08684 1/20 0.34
CDK4 P11802 1/20 0.34
CCNA2 P20248 1/20 0.34
CCND1 P24385 1/20 0.34
CDK2 P24941 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984798 0.79 CA1 (1.00) CA1CA2CA7CA9CA4
SCHEMBL11814244 0.77 CA1 (0.40) CA1CA2CA7CA9EPHX2
SCHEMBL12326178 0.64 ACHE (0.44) CA9ALDH1A1CYP3A4
SCHEMBL3070529 0.63 L3MBTL1 (0.48) CA1CA2CA7CA9EPHX2
SCHEMBL11814298 0.63 ALDH1A1 (0.36) CA1CA2CA7CA9ALDH1A1
SCHEMBL24756167 0.62 CA1 (0.61) CA1CA2CA7CA9CA4
SCHEMBL16071623 0.62 ACHE (0.52) CA1CA2CA7CA9CA4
SCHEMBL11387445 0.62 ABCB1 (0.40) CA1CA2CA7CA9EPHX2
SCHEMBL14390487 0.62 KDM4E (0.55) ALDH1A1MAPK1RECQL
SCHEMBL4395035 0.62 CA1 (1.00) CA1CA2CA7CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO claimed
WO-2001079209-A2 DIAZAFLUORENONE IL-8 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2001-10-25 WO disclosed