SCHEMBL8002294

SCHEMBL8002294

COC(=O)c1cc(C(=O)OC)cc(N(S(=O)(=O)/C=C/c2cccc(Cl)c2)S(=O)(=O)/C=C/c2cccc(Cl)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 4/20 0.46
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAOB P27338 2/20 0.40
MAOA P21397 1/20 0.40
RELA Q04206 1/20 0.39
PTGES2 Q9H7Z7 3/20 0.39
P4HB P07237 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NR1H4 Q96RI1 1/20 0.38
AKR1C3 P42330 1/20 0.37
FBP1 P09467 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8001587 0.88 ALDH1A1 (0.45) NFE2L2MAPTSMN1; SMN2CYP1A2CYP2C9
SCHEMBL8004163 0.87 TSHR (0.42) NFE2L2MAPTNPC1POLBRAB9A
SCHEMBL7998337 0.81 NFE2L2 (0.62) NFE2L2CYP1A2CYP2C9RELAPTGES2
SCHEMBL7990203 0.80 NFE2L2 (0.47) NFE2L2CYP1A2CYP2C9MAOBMAOA
SCHEMBL7988658 0.80 PPARG (0.44) MAPTNPC1POLBRAB9ACYP1A2
SCHEMBL7998331 0.78 NFE2L2 (0.48) NFE2L2MAPTSMN1; SMN2CYP1A2CYP2C9
SCHEMBL7998940 0.77 NFE2L2 (0.64) NFE2L2RELAFBP1
SCHEMBL7988661 0.75 PPARG (0.49) NFE2L2MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL8002291 0.75 NFE2L2 (0.60) NFE2L2RELAFBP1
SCHEMBL7998895 0.73 NFE2L2 (0.41) NFE2L2CYP1A2CYP2C9PTGES2FBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009120783-A1 HIGH AFFINITY INHIBITORS OF HEPATITIS C VIRUS NS3/4A PROTEASE THE JOHNS HOPKINS UNIVERSITY (US) 2009-10-01 WO disclosed