SCHEMBL8003097

SCHEMBL8003097

N#CC1(c2ccccn2)CCN(CCC(N)=O)CC1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.56
PRKCA P17252 1/20 0.51
PTPN2 P17706 1/20 0.51
HTR7 P34969 1/20 0.51
CCR1 P32246 1/20 0.45
CHRM1 P11229 1/20 0.44
KCNH2 Q12809 1/20 0.42
ADRA1D P25100 1/20 0.40
ADRA1B P35368 1/20 0.40
OPRM1 P35372 2/20 0.39
SPR P35270 1/20 0.39
HTR1A P08908 2/20 0.39
HSD11B1 P28845 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
OPRD1 P41143 1/20 0.38
F11 P03951 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7930702 0.81 ADRA1A (0.56) ADRA1APRKCAPTPN2HTR7CCR1
SCHEMBL8004598 0.81 ADRA1A (0.53) ADRA1APRKCAPTPN2HTR7CCR1
SCHEMBL16549656 0.81 ADRA1A (0.55) ADRA1APRKCAPTPN2HTR7CCR1
SCHEMBL6887265 0.78 ADRA1A (0.52) ADRA1APRKCAPTPN2HTR7CCR1
SCHEMBL7662399 0.78 ADRA1A (0.45) ADRA1AADRA1DADRA1BOPRM1
SCHEMBL761722 0.77 PRKCA (0.51) ADRA1APRKCAPTPN2HTR7CCR1
SCHEMBL7668741 0.77 ADRA1A (0.44) ADRA1AADRA1DADRA1BOPRM1
Hydrochloric Acid SCHEMBL7664053 0.77 ADRA1A (0.44) ADRA1AADRA1DADRA1BOPRM1
SCHEMBL3323620 0.76 OPRM1 (0.50) ADRA1APRKCAPTPN2HTR7OPRM1
Hydrochloric Acid SCHEMBL7664114 0.76 ADRA1A (0.44) ADRA1AADRA1DADRA1BOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000025782-A1 DIHYDROPYRIDINONES AND PYRROLINONES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-11 WO disclosed