SCHEMBL8008384

SCHEMBL8008384

COc1ccc2c(N)cc(-c3nc(C4CC4)cs3)nc2c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.36
KDM4E B2RXH2 4/20 0.36
FPR2 P25090 2/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
C1S P09871 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 3/20 0.32
MAPT P10636 3/20 0.32
RAB9A P51151 3/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
HPGD P15428 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
G6PD P11413 1/20 0.32
LMNA P02545 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15216098 0.96 C1S (0.37) ALDH1A1KDM4EFPR2GABRA1GABRG2
SCHEMBL3672299 0.89 FPR2 (0.36) ALDH1A1KDM4EFPR2GABRA1GABRG2
SCHEMBL3675051 0.87 FPR2 (0.37) ALDH1A1KDM4EFPR2GABRA1GABRG2
SCHEMBL8005668 0.85 C1S (0.36) ALDH1A1KDM4EFPR2GABRA1GABRG2
SCHEMBL8005137 0.84 KDM4E (0.39) ALDH1A1KDM4ENPC1MAPTRAB9A
SCHEMBL8006162 0.81 ALDH1A1 (0.37) ALDH1A1KDM4EC1STDP1NPC1
SCHEMBL8003756 0.80 KDM4E (0.36) ALDH1A1KDM4ENPC1MAPTRAB9A
SCHEMBL8005422 0.80 ALDH1A1 (0.36) ALDH1A1KDM4ETDP1NPC1MAPT
SCHEMBL8006048 0.80 KDM4E (0.36) ALDH1A1KDM4ENPC1MAPTRAB9A
SCHEMBL8003492 0.80 KDM4E (0.36) ALDH1A1KDM4ETDP1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2250174-B1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS INC (US) 2013-08-28 EP disclosed
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed