SCHEMBL8003824

SCHEMBL8003824

CC(C)c1ccc(C2(N)CCC(=O)CC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.39
TYR P14679 2/20 0.38
HSD11B1 P28845 2/20 0.38
CYP19A1 P11511 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C9 P11712 1/20 0.36
POLB P06746 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
MYC P01106 1/20 0.36
MAX P61244 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1719333 0.85 TYR (0.41) PIM1TYR
SCHEMBL10132207 0.79 MEN1 (0.39) HSD11B1MEN1KMT2ACYP2C9
SCHEMBL11793971 0.79 TYR (0.40) PIM1TYRHSD11B1MEN1KMT2A
Hydrochloric Acid SCHEMBL5671167 0.78
SCHEMBL11800670 0.76 ALOX5 (0.42) PIM1TYRHSD11B1MEN1KMT2A
SCHEMBL7991720 0.76 HSD11B1 (0.44) PIM1HSD11B1MEN1KMT2ACYP2C9
SCHEMBL8005872 0.76 MAOB (0.39) HSD11B1MEN1KMT2ACYP2C9SLC6A3
SCHEMBL612898 0.75 MAOB (0.43) PIM1HSD11B1POLBRAB9ASLC6A4
SCHEMBL29218720 0.75 OPRL1 (0.39) TYRRAB9A
SCHEMBL614021 0.75 MEN1 (0.63) MEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009156100-A1 SUBSTITUTED ISOQUINOLINES AND ISOQUINOLINONES AS RHO KINASE INHIBITORS SANOFI-AVENTIS (FR) 2009-12-30 WO disclosed