SCHEMBL8003967

SCHEMBL8003967

[CH2]CCN1CCC(c2ccccn2)CC1

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 16/20 0.52
DRD2 P14416 10/20 0.51
DRD3 P35462 7/20 0.50
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
CHRM2 P08172 1/20 0.42
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7833509 0.84 DRD2 (0.59) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL21274017 0.83 DRD4 (0.50) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL6196064 0.82 DRD4 (0.52) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL6198971 0.82 ADRA1D (0.55) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL10819399 0.81 DRD4 (0.54) DRD4DRD2DRD3ADRA1DADRA1A
Hydrochloric Acid SCHEMBL7660487 0.81 DRD4 (0.51) DRD4DRD2DRD3ADRA1DADRA1A
Hydrochloric Acid SCHEMBL8181520 0.81 DRD4 (0.51) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL7212038 0.79 DRD4 (0.59) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL6198252 0.79 ADRA1D (0.49) DRD4DRD2DRD3ADRA1DADRA1A
SCHEMBL6198244 0.79 ADRA1A (0.60) DRD4DRD2DRD3ADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000025782-A1 DIHYDROPYRIDINONES AND PYRROLINONES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-05-11 WO disclosed