SCHEMBL7995599

SCHEMBL7995599

CS(=O)(=O)c1cc(COC(=O)NC(=N)N)ccc1Oc1ccc2ncccc2c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
SCN9A Q15858 1/20 0.40
BRD4 O60885 1/20 0.37
PPARG P37231 2/20 0.36
PTGER3 P43115 2/20 0.36
GCK P35557 2/20 0.36
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
ROCK2 O75116 1/20 0.35
ALOX5 P09917 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ABL1 P00519 1/20 0.34
AXL P30530 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8101760 0.99 ALDH1A1 (0.41) ALDH1A1SCN9ABRD4PPARGPTGER3
Hydrochloric Acid SCHEMBL8007030 0.99 ALDH1A1 (0.41) ALDH1A1SCN9ABRD4PPARGPTGER3
SCHEMBL7995604 0.85 AOC3 (0.40) ALDH1A1SCN9ABRD4PPARG
Hydrochloric Acid SCHEMBL8104379 0.84 AOC3 (0.41) ALDH1A1SCN9ABRD4PPARG
Hydrochloric Acid SCHEMBL8007034 0.84 AOC3 (0.41) ALDH1A1SCN9ABRD4PPARG
SCHEMBL8831746 0.83 PLK1 (0.47) ALDH1A1SCN9ABRD4PTGER3CYP3A4
Water SCHEMBL8095247 0.82 SCN9A (0.40) ALDH1A1SCN9ABRD4PPARGPTGER3
SCHEMBL8004004 0.81 KCNQ3 (0.39)
SCHEMBL8004732 0.75 ALOX15 (0.62) ALDH1A1SCN9ABRD4PPARGPTGER3
SCHEMBL8005829 0.71 PPARG (0.37) SCN9APPARGGCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP disclosed
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed
EP-0748795-A2 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-12-18 EP disclosed