SCHEMBL8006015

SCHEMBL8006015

CCOC(=O)CCCN1C(=O)c2ccc(N)cc2C1=O

nearest known ligand 0.72

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 4/20 0.72
CASP1 P29466 2/20 0.72
MAPT P10636 2/20 0.72
ALOX15 P16050 1/20 0.72
CASP7 P55210 1/20 0.72
KMT2A Q03164 4/20 0.67
MEN1 O00255 3/20 0.67
GAA P10253 1/20 0.67
TNF P01375 4/20 0.60
ALDH1A1 P00352 5/20 0.50
TSHR P16473 1/20 0.50
MAPK1 P28482 1/20 0.50
PIN1 Q13526 1/20 0.48
PIN4 Q9Y237 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL523511 0.84 PIN1 (0.68) HSD17B10CASP1MAPTALOX15CASP7
SCHEMBL7424373 0.84 KMT2A (0.63) HSD17B10MAPTKMT2AMEN1TNF
SCHEMBL3862952 0.84 TNF (0.51) HSD17B10CASP1MAPTALOX15CASP7
SCHEMBL918351 0.82 HDAC3 (0.56) HSD17B10CASP1MAPTALOX15CASP7
SCHEMBL25358575 0.81 HSD17B10 (1.00) HSD17B10CASP1MAPTALOX15CASP7
SCHEMBL9798967 0.80 ALDH1A1 (0.58) HSD17B10MAPTKMT2AMEN1ALDH1A1
SCHEMBL2651666 0.79 HSD17B10 (0.66) HSD17B10CASP1MAPTALOX15CASP7
SCHEMBL7589770 0.79 HDAC8 (0.59) HSD17B10MAPTKMT2AMEN1GAA
SCHEMBL7549194 0.79 HDAC8 (0.59) HSD17B10MAPTKMT2AMEN1GAA
SCHEMBL2618100 0.79 HDAC8 (0.59) HSD17B10MAPTKMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed
WO-1999051590-A1 SUBSTITUTED INDOLINONES AS KINASE INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-14 WO disclosed