SCHEMBL8006531

SCHEMBL8006531

N#Cc1c(N)nc(SCc2ccccn2)c(C#N)c1-c1ccc(C[C@H]2CCCC[C@@H]2O)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
PKM P14618 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
ADORA1 P30542 17/20 0.54
ADORA2A P29274 5/20 0.54
ADORA3 P0DMS8 4/20 0.54
ADORA2B P29275 5/20 0.47
SLC6A3 Q01959 1/20 0.45
MEN1 O00255 1/20 0.44
PPARG P37231 1/20 0.44
KMT2A Q03164 1/20 0.44
NCOA2 Q15596 1/20 0.44
NCOA1 Q15788 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
RET P07949 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006044 0.85 ADORA1 (0.65) ALDH1A1SMN1; SMN2ADORA1ADORA2AADORA3
SCHEMBL8006647 0.85 ADORA1 (0.64) ADORA1SLC6A3RET
SCHEMBL12943304 0.84 ADORA1 (0.55) ALDH1A1PKMSMN1; SMN2ADORA1ADORA2A
SCHEMBL8007650 0.83 ADORA1 (0.56) ADORA1SLC6A3RET
SCHEMBL7997244 0.83 ADORA1 (0.64) ADORA1SLC6A3RET
SCHEMBL7997209 0.83 ADORA1 (0.62) ADORA1ADORA3ADORA2B
SCHEMBL8010353 0.83 ADORA1 (0.71) ADORA1SLC6A3MEN1PPARGKMT2A
SCHEMBL8008772 0.82 ADORA1 (0.55) ALDH1A1PKMSMN1; SMN2ADORA1ADORA2A
SCHEMBL8008969 0.81 ADORA1 (0.71) ADORA1SLC6A3RET
SCHEMBL8008967 0.80 ADORA1 (0.52) ALDH1A1ADORA1ADORA2AADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100827-A1 CYCLOALKOXY-SUBSTITUTED 4-PHENYL-3,5-DICYANOPYRIDINES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-08-20 WO disclosed