SCHEMBL8007650

SCHEMBL8007650

Cc1nc(CSc2nc(N)c(C#N)c(-c3ccc(C[C@H]4CCCC[C@@H]4O)cc3)c2C#N)cs1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 19/20 0.56
SLC6A3 Q01959 1/20 0.51
RET P07949 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006647 0.92 ADORA1 (0.64) ADORA1SLC6A3RET
SCHEMBL7997244 0.90 ADORA1 (0.64) ADORA1SLC6A3RET
SCHEMBL8010353 0.89 ADORA1 (0.71) ADORA1SLC6A3RET
SCHEMBL8008969 0.88 ADORA1 (0.71) ADORA1SLC6A3RET
SCHEMBL12943379 0.85 ADORA1 (0.61) ADORA1SLC6A3
SCHEMBL8006531 0.83 ALDH1A1 (0.54) ADORA1SLC6A3RET
SCHEMBL8008774 0.83 ADORA1 (0.54) ADORA1SLC6A3
SCHEMBL7997209 0.82 ADORA1 (0.62) ADORA1
SCHEMBL13929772 0.81 ADORA1 (0.63) ADORA1SLC6A3RET
SCHEMBL8008967 0.80 ADORA1 (0.52) ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100827-A1 CYCLOALKOXY-SUBSTITUTED 4-PHENYL-3,5-DICYANOPYRIDINES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-08-20 WO disclosed