SCHEMBL8008967

SCHEMBL8008967

COCCSc1nc(N)c(C#N)c(-c2ccc(C[C@H]3CCCC[C@@H]3O)cc2)c1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 12/20 0.52
NPSR1 Q6W5P4 3/20 0.48
KDM4E B2RXH2 2/20 0.48
HTT P42858 1/20 0.48
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PPARG P37231 1/20 0.46
NCOA2 Q15596 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
ADORA2B P29275 4/20 0.45
HTR1B P28222 1/20 0.45
OPRK1 P41145 1/20 0.45
FFAR4 Q5NUL3 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
ADORA2A P29274 1/20 0.45
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997209 0.89 ADORA1 (0.62) ADORA1ADORA2BADORA3
SCHEMBL12943227 0.84 ADORA1 (0.57) ADORA1NPSR1KDM4EHTTALDH1A1
SCHEMBL8007650 0.80 ADORA1 (0.56) ADORA1
SCHEMBL8006044 0.80 ADORA1 (0.65) ADORA1NPSR1KDM4EALDH1A1MEN1
SCHEMBL8006531 0.80 ALDH1A1 (0.54) ADORA1NPSR1ALDH1A1MEN1KMT2A
SCHEMBL8006647 0.80 ADORA1 (0.64) ADORA1
SCHEMBL7997244 0.78 ADORA1 (0.64) ADORA1
SCHEMBL8010353 0.78 ADORA1 (0.71) ADORA1NPSR1MEN1KMT2APPARG
SCHEMBL13914391 0.78 ADORA2B (0.73) ADORA1NPSR1KDM4EHTTALDH1A1
SCHEMBL13914403 0.77 ADORA1 (0.72) ADORA1NPSR1KDM4EHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100827-A1 CYCLOALKOXY-SUBSTITUTED 4-PHENYL-3,5-DICYANOPYRIDINES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-08-20 WO disclosed