SCHEMBL8007057

SCHEMBL8007057

COc1ccc(OC)c(C2C[C@]3(C)[C@H]4CC[C@]5(C)CCC[C@H]5[C@@H]4CC[C@H]3N(C)C2=O)c1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 2/20 0.37
GAA P10253 2/20 0.36
LMNA P02545 2/20 0.36
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
ALDH1A1 P00352 4/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
STS P08842 1/20 0.34
MBOAT4 Q96T53 2/20 0.34
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8018783 0.88 SRD5A1 (0.36) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8018769 0.86 SRD5A1 (0.41) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8024003 0.85 DDB1 (0.41) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8016913 0.83 SRD5A1 (0.43) SRD5A1
SCHEMBL8016758 0.83 MBOAT4 (0.37) CDK5CDK5R1MBOAT4
SCHEMBL8007078 0.79 CDK5 (0.38) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8023771 0.77 SRD5A1 (0.36) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8019107 0.75 CDK5 (0.37) CDK5CDK5R1MBOAT4
SCHEMBL8076029 0.73 NR1I3 (0.47) CDK5CDK5R1
SCHEMBL8018781 0.72 MAPT (0.38) SRD5A1GAALMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed