SCHEMBL8024003

SCHEMBL8024003

COc1cccc(C2C[C@]3(C)[C@H]4CC[C@]5(C)CCC[C@H]5[C@@H]4CC[C@H]3N(C)C2=O)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
SRD5A1 P18405 2/20 0.39
CHRNA7 P36544 2/20 0.36
HSD11B1 P28845 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
GID4 Q8IVV7 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
KMT2A Q03164 1/20 0.34
MBOAT4 Q96T53 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8018769 0.89 SRD5A1 (0.41) DDB1CRBNSRD5A1CDK5CDK5R1
SCHEMBL8007057 0.85 SRD5A1 (0.37) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8016758 0.83 MBOAT4 (0.37) CDK5CDK5R1MBOAT4
SCHEMBL8018783 0.81 SRD5A1 (0.36) SRD5A1CHRNA7HSD11B1CDK5CDK5R1
SCHEMBL8006579 0.81 DDB1 (0.46) DDB1CRBNSRD5A1GID4MEN1
SCHEMBL8019107 0.79 CDK5 (0.37) CDK5CDK5R1MBOAT4
SCHEMBL8007078 0.78 CDK5 (0.38) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8023771 0.78 SRD5A1 (0.36) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8076029 0.74 NR1I3 (0.47) CDK5CDK5R1
SCHEMBL8679342 0.72 SRD5A1 (0.37) SRD5A1CDK5CDK5R1MBOAT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed