SCHEMBL8018783

SCHEMBL8018783

COc1ccccc1C1C[C@]2(C)[C@H]3CC[C@]4(C)CCC[C@H]4[C@@H]3CC[C@H]2N(C)C1=O

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 2/20 0.36
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
MBOAT4 Q96T53 1/20 0.35
SRD5A2 P31213 1/20 0.34
CYP19A1 P11511 3/20 0.34
HSD11B1 P28845 2/20 0.34
NR1I3 Q14994 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007057 0.88 SRD5A1 (0.37) SRD5A1CDK5CDK5R1MBOAT4
SCHEMBL8007078 0.87 CDK5 (0.38) SRD5A1CDK5CDK5R1MBOAT4SRD5A2
SCHEMBL8023771 0.85 SRD5A1 (0.36) SRD5A1CDK5CDK5R1MBOAT4SRD5A2
SCHEMBL8016758 0.83 MBOAT4 (0.37) CDK5CDK5R1MBOAT4CYP19A1NR1I3
SCHEMBL8018769 0.83 SRD5A1 (0.41) SRD5A1CDK5CDK5R1MBOAT4CYP19A1
SCHEMBL8024003 0.81 DDB1 (0.41) SRD5A1CDK5CDK5R1MBOAT4HSD11B1
SCHEMBL8023088 0.80 SRD5A1 (0.39) SRD5A1CDK5CDK5R1MBOAT4SRD5A2
SCHEMBL8679342 0.77 SRD5A1 (0.37) SRD5A1CDK5CDK5R1MBOAT4SRD5A2
SCHEMBL8019107 0.77 CDK5 (0.37) CDK5CDK5R1MBOAT4CYP19A1NR1I3
SCHEMBL8076029 0.75 NR1I3 (0.47) CDK5CDK5R1CYP19A1NR1I3GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0664812-B1 17-BETA-ARYL ESTER CARBOXYLATES OF 4-AZA-5-ALPHA-ANDROSTANE-3-ONES MERCK & CO INC (US) 2000-01-05 EP claimed