SCHEMBL8007497

SCHEMBL8007497

CC1(C)CC(O)CC(C#N)(c2ccccc2)C1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.43
OPRL1 P41146 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
OPRM1 P35372 1/20 0.37
CYP2D6 P10635 1/20 0.34
HSD11B1 P28845 1/20 0.34
CCR2 P41597 1/20 0.34
MAOB P27338 3/20 0.33
MAOA P21397 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097375 0.85 OPRL1 (0.46) OPRD1OPRL1CA12CA1CA2
SCHEMBL8104825 0.79 OPRM1 (0.45) OPRD1OPRL1CA12CA1CA2
SCHEMBL13887044 0.79 MEN1 (0.46) OPRD1OPRL1CA12CA1CA2
SCHEMBL1558648 0.75 MEN1 (0.51) OPRD1OPRL1CA12CA1CA2
SCHEMBL1558649 0.75 MEN1 (0.51) OPRD1OPRL1CA12CA1CA2
SCHEMBL11703497 0.73 MEN1 (0.43) OPRD1OPRL1CA12CA1CA2
SCHEMBL8107113 0.71 OPRL1 (0.46) OPRD1OPRL1CA12CA1CA2
SCHEMBL14491853 0.70 KDM1A (0.47) OPRD1OPRL1KMT2AOPRM1HSD11B1
SCHEMBL17985301 0.70 KDM1A (0.47) OPRD1OPRL1KMT2AOPRM1HSD11B1
SCHEMBL8007148 0.70 OPRM1 (0.38) OPRD1OPRL1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6060484-A Anti-viral method ELI LILLY AND COMPANY (US) 2000-05-09 US disclosed
WO-1997041846-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1997-11-13 WO disclosed
EP-0806205-A2 Urea, thiourea and guanidine compounds and their use as anti-viral agents ELI LILLY AND COMPANY (US) 1997-11-12 EP disclosed