SCHEMBL8007148

SCHEMBL8007148

CC1(C)CC(=O)CC(C#N)(c2ccccc2)C1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.38
OPRD1 P41143 1/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
OPRL1 P41146 1/20 0.35
ALDH1A1 P00352 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MGAT2 Q10469 1/20 0.34
CYP2C9 P11712 1/20 0.33
CYP2D6 P10635 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097373 0.84 OPRM1 (0.45) OPRM1OPRD1CA12CA1CA2
SCHEMBL8104825 0.81 OPRM1 (0.45) OPRM1OPRD1CA12CA1CA2
SCHEMBL13163312 0.75 MEN1 (0.48) OPRM1OPRD1CA12CA1CA2
SCHEMBL11473105 0.74 ALDH1A1 (0.39) MEN1KMT2AALDH1A1NPC1RAB9A
SCHEMBL5370161 0.72 MEN1 (0.43) OPRM1OPRD1CA12CA1CA2
SCHEMBL735798 0.70 MEN1 (0.57) OPRM1OPRD1CA12CA1CA2
SCHEMBL8007497 0.70 OPRD1 (0.43) OPRM1OPRD1CA12CA1CA2
SCHEMBL647137 0.69 CTSK (0.36) ALDH1A1
SCHEMBL432561 0.68 OPRM1 (0.59) OPRM1OPRD1CA12CA1CA2
Ethylene SCHEMBL3968375 0.68 MEN1 (0.53) OPRM1OPRD1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6060484-A Anti-viral method ELI LILLY AND COMPANY (US) 2000-05-09 US disclosed
WO-1997041846-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1997-11-13 WO disclosed
EP-0806205-A2 Urea, thiourea and guanidine compounds and their use as anti-viral agents ELI LILLY AND COMPANY (US) 1997-11-12 EP disclosed