SCHEMBL8007547

SCHEMBL8007547

NCCCn1ncc2ccc(I)cc21

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.55
HTR2C P28335 5/20 0.55
HTR2B P41595 4/20 0.55
KMO O15229 10/20 0.45
HTR1A P08908 2/20 0.38
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
HTR1D P28221 1/20 0.38
HTR7 P34969 1/20 0.38
HTR4 Q13639 1/20 0.38
CYP1A2 P05177 1/20 0.36
SYK P43405 1/20 0.34
P2RX7 Q99572 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6741175 0.81 HTR2A (0.46) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL3779615 0.81 KMO (0.42) HTR2AHTR2CHTR2BKMOHTR1A
Ammonia Solution, Strong SCHEMBL8009916 0.79 HTR2A (0.45) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL8013345 0.79 HTR2A (0.52) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL3784975 0.79 CHRM2 (0.41) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL3777872 0.77 HTR2A (0.40) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL3243999 0.77 CYP1A2 (0.58) HTR2AHTR2CHTR2BKMOADRA2A
SCHEMBL4539220 0.76 MCHR1 (0.47) HTR2AHTR2CHTR2B
SCHEMBL3784965 0.76 HTR2A (0.42) HTR2AHTR2CHTR2BKMOHTR1A
SCHEMBL8007092 0.75 HTR2C (0.48) HTR2AHTR2CHTR2BKMOHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000017170-A2 N1-SUBSTITUTED BENZOPYRAZOLES AS INHIBITORS OF 5-HT2 RECEPTORS VERNALIS RESEARCH LIMITED (GB) 2000-03-30 WO disclosed