SCHEMBL8007749

SCHEMBL8007749

Cc1nnc(CCCCc2cccc(-c3nn(C)nc3-c3ccccc3)c2)o1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.39
HSD11B1 P28845 2/20 0.37
GRIN1 Q05586 3/20 0.36
GRIN2B Q13224 3/20 0.36
KDM4E B2RXH2 1/20 0.35
THRB P10828 1/20 0.35
KMT2A Q03164 2/20 0.34
GLS O94925 1/20 0.34
RAB9A P51151 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
PKM P14618 1/20 0.34
STAT1 P42224 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007765 0.99 POLB (0.38) POLBHSD11B1GRIN1GRIN2BKDM4E
SCHEMBL8008284 0.99 POLB (0.38) POLBHSD11B1GRIN1GRIN2BKDM4E
SCHEMBL8010417 0.98 POLB (0.41) POLBHSD11B1GRIN1GRIN2BKMT2A
SCHEMBL8013957 0.87 GRIN1 (0.36) POLBHSD11B1GRIN1GRIN2B
SCHEMBL8007717 0.82 HDAC6 (0.33) GRIN1GRIN2B
SCHEMBL7998525 0.81 HDAC1 (0.33) POLBGRIN1GRIN2BKDM4E
SCHEMBL7999089 0.78 HDAC1 (0.34) GRIN1GRIN2BKDM4E
SCHEMBL10260440 0.76 ATM (0.36) POLBKDM4EKMT2ARAB9ANPC1
SCHEMBL8007763 0.75 GRIN1 (0.35) GRIN1GRIN2BKDM4ERAB9ANPC1
SCHEMBL10261621 0.75 ATM (0.36) POLBKDM4EKMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed