SCHEMBL8007717

SCHEMBL8007717

Cc1nnc(CCCC/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)o1

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.33
HDAC1 Q13547 5/20 0.33
HDAC8 Q9BY41 4/20 0.33
GRIN1 Q05586 4/20 0.33
GRIN2B Q13224 4/20 0.33
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
SIGMAR1 Q99720 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7998525 0.97 HDAC1 (0.33) HDAC6HDAC1HDAC8GRIN1GRIN2B
SCHEMBL7999089 0.93 HDAC1 (0.34) HDAC6HDAC1HDAC8GRIN1GRIN2B
SCHEMBL8007763 0.86 GRIN1 (0.35) HDAC6HDAC1HDAC8GRIN1GRIN2B
SCHEMBL8007749 0.82 POLB (0.39) GRIN1GRIN2B
SCHEMBL7998527 0.81 GRIN1 (0.35) HDAC6HDAC1HDAC8GRIN1GRIN2B
SCHEMBL8007765 0.81 POLB (0.38) GRIN1GRIN2B
SCHEMBL8008284 0.81 POLB (0.38) GRIN1GRIN2B
SCHEMBL8010417 0.80 POLB (0.41) GRIN1GRIN2BTDP1
SCHEMBL7998444 0.80 L3MBTL1 (0.32) HDAC6HDAC1HDAC8
SCHEMBL10293079 0.79 FAAH (0.30) HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed