SCHEMBL7998525

SCHEMBL7998525

Cc1nnc(CCC/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)o1

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 6/20 0.33
HDAC8 Q9BY41 6/20 0.33
HDAC6 Q9UBN7 6/20 0.33
GRIN1 Q05586 4/20 0.33
GRIN2B Q13224 4/20 0.33
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
SIGMAR1 Q99720 2/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
TSHR P16473 1/20 0.30
XBP1 P17861 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8007717 0.97 HDAC6 (0.33) HDAC1HDAC8HDAC6GRIN1GRIN2B
SCHEMBL7999089 0.94 HDAC1 (0.34) HDAC1HDAC8HDAC6GRIN1GRIN2B
SCHEMBL8007763 0.87 GRIN1 (0.35) HDAC1HDAC8HDAC6GRIN1GRIN2B
SCHEMBL7998527 0.82 GRIN1 (0.35) HDAC1HDAC8HDAC6GRIN1GRIN2B
SCHEMBL8007749 0.81 POLB (0.39) GRIN1GRIN2BKDM4EPOLB
SCHEMBL8010417 0.81 POLB (0.41) GRIN1GRIN2BTDP1POLB
SCHEMBL8008284 0.80 POLB (0.38) GRIN1GRIN2BKDM4EPOLB
SCHEMBL8007765 0.80 POLB (0.38) GRIN1GRIN2BKDM4EPOLB
SCHEMBL7998577 0.79 L3MBTL1 (0.32) HDAC1HDAC8HDAC6ALDH1A1GAA
SCHEMBL10293080 0.79 CYP1A2 (0.31) ALDH1A1KDM4EUSP2TSHRXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed