SCHEMBL8007763

SCHEMBL8007763

Cc1nnc(C/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)o1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 5/20 0.35
GRIN2B Q13224 5/20 0.35
HDAC1 Q13547 3/20 0.33
HDAC8 Q9BY41 3/20 0.33
HDAC6 Q9UBN7 3/20 0.33
DCTPP1 Q9H773 1/20 0.32
TSHR P16473 3/20 0.32
MAPK1 P28482 2/20 0.32
HSD17B10 Q99714 2/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
XBP1 P17861 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NPC1 O15118 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGS1 P23219 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7999089 0.89 HDAC1 (0.34) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL7998525 0.87 HDAC1 (0.33) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL8007717 0.86 HDAC6 (0.33) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL7998527 0.86 GRIN1 (0.35) GRIN1GRIN2BHDAC1HDAC8HDAC6
SCHEMBL4191955 0.79 HTR2A (0.39) TSHRALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL10260657 0.77 CYP1A2 (0.32) HDAC6PPARGPPARA
SCHEMBL8001035 0.77 L3MBTL1 (0.34) HDAC1HDAC8HDAC6ALDH1A1KDM4E
SCHEMBL10292814 0.77 CYP1A2 (0.32) TSHRMAPK1HSD17B10ALDH1A1KDM4E
SCHEMBL8007749 0.75 POLB (0.39) GRIN1GRIN2BKDM4ENPC1RAB9A
SCHEMBL8010417 0.75 POLB (0.41) GRIN1GRIN2BNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed