SCHEMBL8007795

SCHEMBL8007795

COc1ccc(-c2cccc(-c3cocn3)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.54
ABCB1 P08183 2/20 0.54
BCR P11274 2/20 0.54
SCN9A Q15858 2/20 0.49
ENPP3 O14638 2/20 0.44
ENPP1 P22413 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
RAB9A P51151 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
DYRK1A Q13627 2/20 0.44
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2E1 P05181 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2A6 P11509 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3635892 0.86 DYRK1A (0.53) SCN9ARAB9AKMT2ADYRK1ACYP1A2
SCHEMBL1186835 0.85 ENPP3 (0.50) ENPP3ENPP1RAB9AMEN1KMT2A
SCHEMBL16159336 0.82 SCN9A (0.55) SCN9AENPP3HDAC4CYP1A1CYP1A2
SCHEMBL14564377 0.82 SCN9A (0.62) SCN9AHDAC4
SCHEMBL8007463 0.80 ESR1 (0.57) ABL1ABCB1BCRSCN9AMEN1
SCHEMBL1180429 0.78 ABL1 (0.83) ABL1ABCB1BCRHDAC4HDAC2
SCHEMBL16159397 0.77 SCN9A (0.54) SCN9AHDAC4
SCHEMBL28428427 0.75 ABL1 (0.57) ABL1ABCB1BCRRAB9ADYRK1A
SCHEMBL16159400 0.75 SCN9A (0.55) SCN9AHDAC4
SCHEMBL16159804 0.75 SCN9A (0.51) SCN9AHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000019994-A9 ESTROGEN RECEPTOR LIGANDS UNIV ILLINOIS (US) 2000-08-31 WO disclosed
WO-2000019994-A1 ESTROGEN RECEPTOR LIGANDS BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2000-04-13 WO disclosed