SCHEMBL8007463

SCHEMBL8007463

Oc1ccc(-c2cccc(-c3cocn3)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.57
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
SCN9A Q15858 2/20 0.52
ABL1 P00519 2/20 0.50
ABCB1 P08183 2/20 0.50
BCR P11274 2/20 0.50
HSD17B1 P14061 7/20 0.48
HSD17B2 P37059 7/20 0.48
ESR2 Q92731 1/20 0.44
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 2/20 0.41
MMP3 P08254 1/20 0.41
BCL2L1 Q07817 1/20 0.41
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DUSP3 P51452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14564377 0.86 SCN9A (0.62) SCN9A
SCHEMBL4751198 0.84 HSD17B1 (0.58) SCN9AHSD17B1HSD17B2CYP3A4CYP2C9
SCHEMBL1186172 0.84 ESR1 (0.46) ESR1MEN1KMT2ASCN9AHSD17B1
SCHEMBL16159336 0.83 SCN9A (0.55) ESR1SCN9AHSD17B1HSD17B2ESR2
SCHEMBL16159397 0.81 SCN9A (0.54) SCN9A
SCHEMBL8007795 0.80 ABL1 (0.54) MEN1KMT2ASCN9AABL1ABCB1
SCHEMBL16159400 0.79 SCN9A (0.55) SCN9AHSD17B1HSD17B2
SCHEMBL16159398 0.77 SCN9A (0.52) ESR1SCN9AHSD17B1HSD17B2ESR2
SCHEMBL27607302 0.76 HDAC4 (0.51) MEN1KMT2ASCN9AALDH1A1MAPT
SCHEMBL16159195 0.76 SCN9A (0.49) SCN9ADUSP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000019994-A9 ESTROGEN RECEPTOR LIGANDS UNIV ILLINOIS (US) 2000-08-31 WO disclosed
WO-2000019994-A1 ESTROGEN RECEPTOR LIGANDS BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2000-04-13 WO disclosed